SCHEMBL2295993

SCHEMBL2295993

O=C(O)c1cnn(-c2ncccc2Cl)c1C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.59
MAPT P10636 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CRHBP P24387 1/20 0.47
MC4R P32245 1/20 0.47
CRHR2 Q13324 1/20 0.47
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
MALT1 Q9UDY8 11/20 0.46
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
KEAP1 Q14145 3/20 0.44
NFE2L2 Q16236 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31377061 1.00 POLB (0.59) POLBMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL31377060 0.90 POLB (0.46) POLBMAPTSMN1; SMN2MALT1KDM4E
SCHEMBL31007079 0.90 POLB (0.46) POLBMAPTSMN1; SMN2MALT1KDM4E
SCHEMBL30097595 0.89 MALT1 (0.45) POLBMAPTSMN1; SMN2MALT1KDM4E
SCHEMBL30097896 0.87 POLB (0.62) POLBMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL27171661 0.87 POLB (0.62) POLBMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL30861257 0.86 POLB (0.60) POLBMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL27171662 0.86 POLB (0.60) POLBMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL21605010 0.85 MAPT (0.59) POLBMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL21605033 0.85 MAPT (0.56) POLBMAPTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240425480-A1 NOVEL PYRIDINE DERIVATIVE COMPOUND AS RON INHIBITOR LG CHEM, LTD. (KR) 2024-12-26 US disclosed
US-20240317739-A1 NOVEL UREA DERIVATIVE COMPOUND AS RON INHIBITOR LG CHEM, LTD. (KR) 2024-09-26 US disclosed
WO-2024134514-A1 NOVEL COMPOUND AS RON INHIBITOR 주식회사 엘지화학 2024-06-27 WO disclosed
EP-4349825-A1 NOVEL PYRIDINE DERIVATIVE COMPOUND AS RON INHIBITOR LG Chem, Ltd. (KR) 2024-04-10 EP disclosed
EP-4339196-A1 NOVEL UREA DERIVATIVE COMPOUND AS RON INHIBITOR LG Chem, Ltd. (KR) 2024-03-20 EP disclosed
CN-117500804-A Novel urea derivative compounds as RON inhibitors 株式会社LG化学 2024-02-02 CN disclosed
CN-117396468-A Novel pyridine derivative compounds as RON inhibitors 株式会社LG化学 2024-01-12 CN disclosed
EP-3807266-B1 PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2023-10-25 EP disclosed
EP-3807266-B1 PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2023-10-25 EP disclosed
CN-112585128-B Pyrazole derivatives as MALT1 inhibitors 詹森药业有限公司 2023-02-21 CN disclosed
WO-2019243964-A1 PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2019-12-26 WO disclosed
EP-2462139-B1 SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2015-01-14 EP disclosed
EP-2462139-B1 SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2015-01-14 EP disclosed
US-8399451-B2 Heterocyclic compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2013-03-19 US disclosed
US-8399451-B2 Heterocyclic compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2013-03-19 US disclosed
US-8399451-B2 Heterocyclic compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2013-03-19 US disclosed
US-20110190255-A1 HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2011-08-04 US disclosed
US-20110190255-A1 HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2011-08-04 US disclosed
US-20110190255-A1 HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY 2011-08-04 US disclosed
WO-2011017578-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-02-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190255-A1 HETEROCYCLIC COMPOUNDS S1PR1, S1PR3, S1PR5 POLB 3979/4885MAPT 4760/4885SMN1; SMN2 1771/4885
US-20240425480-A1 NOVEL PYRIDINE DERIVATIVE COMPOUND AS RON INHIBITOR RET, MST1R, ROS1 POLB 4572/4885MAPT 4286/4885SMN1; SMN2 4129/4885
US-20240317739-A1 NOVEL UREA DERIVATIVE COMPOUND AS RON INHIBITOR CDKN1A, RET, UBTF POLB 3957/4885MAPT 2721/4885SMN1; SMN2 4350/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.