SCHEMBL2296677

SCHEMBL2296677

CN(C)c1ccc(-c2ccc(-n3c(CC4CCN(C(=O)C5CC5)C4)n[nH]c3=O)c(F)c2)cc1

nearest known ligand 0.79

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
FASN P49327 20/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2296669 1.00 FASN (0.79) FASN
SCHEMBL2356541 0.91 FASN (0.68) FASN
SCHEMBL2358746 0.91 FASN (0.83) FASN
SCHEMBL2357573 0.90 FASN (0.81) FASN
SCHEMBL2296370 0.90 FASN (0.74) FASN
SCHEMBL2296365 0.90 FASN (0.74) FASN
SCHEMBL2355630 0.89 FASN (0.81) FASN
SCHEMBL12425223 0.89 FASN (0.80) FASN
SCHEMBL2355745 0.89 FASN (0.80) FASN
SCHEMBL2355905 0.89 FASN (1.00) FASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2538787-A1 TRIAZOLONES AS FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline LLC (US) 2013-01-02 EP disclosed
WO-2011103546-A1 TRIAZOLONES AS FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2011-08-25 WO disclosed