SCHEMBL2297180

SCHEMBL2297180

CNC(=O)c1c(-c2ccc(F)cc2)oc2cc(NS(=O)(=O)CCc3ccc(Br)c(C)c3)c(C3CC3)cc12

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.51
CYP2C9 P11712 5/20 0.51
CYP2C19 P33261 4/20 0.51
KCNH2 Q12809 4/20 0.47
CYP2C8 P10632 5/20 0.37
NR1I2 O75469 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2297799 0.93 CYP2C9 (0.55) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2300577 0.91 CYP2C9 (0.50) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2299493 0.91 CYP2C9 (0.49) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2297463 0.89 CYP2C9 (0.52) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2299889 0.89 CYP2C9 (0.48) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2299423 0.89 CYP2C9 (0.54) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2299027 0.88 CYP2C9 (0.50) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2296869 0.88 CYP2C9 (0.49) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL2296858 0.87 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19KCNH2CYP2C8
SCHEMBL2300225 0.87 CYP2C9 (0.47) CYP3A4CYP2C9CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103063-A1 THERAPEUTIC COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-08-25 WO disclosed