SCHEMBL22977477

SCHEMBL22977477

CS(=O)(=O)N1CCC(Nc2ncc(Cl)c(Cl)n2)CC1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 18/20 0.68
CDK2 P24941 18/20 0.68
CDK1 P06493 4/20 0.68
CCNB1 P14635 4/20 0.68
CCNB2 O95067 3/20 0.68
CCNE2 O96020 3/20 0.68
CDK5 Q00535 3/20 0.68
CDK5R1 Q15078 3/20 0.68
CCNB3 Q8WWL7 3/20 0.68
CCND1 P24385 12/20 0.61
CDK6 Q00534 12/20 0.61
CCNT1 O60563 6/20 0.61
CDK4 P11802 6/20 0.61
CDK9 P50750 6/20 0.61
CCND3 P30281 1/20 0.61
IKBKB O14920 1/20 0.59
MAPK3 P27361 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25400997 0.86 CCNE1 (0.61) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL30537253 0.86 CCNE1 (0.61) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL26941919 0.86 CCNE1 (0.62) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL29631625 0.85 CCNE1 (0.55) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL22901115 0.85 CCNE1 (0.55) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL22901105 0.85 CCNE1 (0.65) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL29631651 0.85 CCNE1 (0.65) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL29754817 0.85 IKBKB (0.59) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL30726194 0.82 CCNE1 (0.57) CCNE1CDK2CDK1CCNB1CCNB2
SCHEMBL27033634 0.82 CCNE1 (0.57) CCNE1CDK2CDK1CCNB1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250243183-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION 2025-07-31 US disclosed
US-12312331-B2 Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors INCYTE CORPORATION (US) 2025-05-27 US disclosed
CN-116348458-A Imidazolylpyrimidinylamine compounds as CDK2 inhibitors 因赛特公司 2023-06-27 CN disclosed
US-20230024173-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION 2023-01-26 US disclosed
US-20230024173-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION 2023-01-26 US disclosed
US-11427567-B2 Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors INCYTE CORPORATION (US) 2022-08-30 US disclosed
EP-4013750-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS Incyte Corporation (US) 2022-06-22 EP disclosed
WO-2021030537-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION (US) 2021-02-18 WO disclosed
WO-2021030537-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION (US) 2021-02-18 WO disclosed
US-20210047294-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION 2021-02-18 US disclosed
US-20210047294-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION 2021-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12312331-B2 Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors CDK2, CDK4, CDK2AP2 CCNE1 43/4885CDK2 1/4885CDK1 7/4885
US-11427567-B2 Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors CDK2, CDK4, CDK2AP2 CCNE1 43/4885CDK2 1/4885CDK1 7/4885
US-20210047294-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS CDK2, CDK4, CDK2AP2 CCNE1 43/4885CDK2 1/4885CDK1 7/4885
US-20230024173-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS CDK2, CDK4, CDK2AP2 CCNE1 43/4885CDK2 1/4885CDK1 7/4885
US-20250243183-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS CDK2, CDK4, CDK2AP2 CCNE1 43/4885CDK2 1/4885CDK1 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.