SCHEMBL22979231

SCHEMBL22979231

Cc1ccccc1-c1nc2c3ccccc3nc(N[C@@H]3CNCCNC3=O)n2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
TSHR P16473 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
MAPT P10636 5/20 0.37
POLB P06746 3/20 0.37
CHEK2 O96017 1/20 0.36
TP53 P04637 4/20 0.35
RAD52 P43351 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
THRB P10828 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HCRTR1 O43613 1/20 0.35
HTT P42858 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22981147 1.00 CYP1A2 (0.41) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL29646458 1.00 CYP1A2 (0.41) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL29645938 1.00 CYP1A2 (0.41) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL22979373 1.00 CYP1A2 (0.41) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL29645531 1.00 CYP1A2 (0.41) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL22979391 0.90 CYP1A2 (0.43) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL22979228 0.90 CYP1A2 (0.43) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL22979468 0.90 CYP1A2 (0.43) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL29645753 0.90 CYP1A2 (0.43) CYP1A2HSD17B10CYP3A4CYP2D6TSHR
SCHEMBL29646184 0.90 CYP1A2 (0.43) CYP1A2HSD17B10CYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP claimed
WO-2021028382-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO claimed