SCHEMBL2299146

SCHEMBL2299146

CCCC(NC(=O)c1cncc2c1cnn2-c1ccc(F)cc1)c1cncc(S(=O)(=O)O)c1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.71
CYP3A4 P08684 1/20 0.62
KCNH2 Q12809 2/20 0.50
ADRB1 P08588 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL568461 1.00 CCR1 (0.71) CCR1CYP3A4KCNH2ADRB1
SCHEMBL568695 0.93 CCR1 (0.76) CCR1CYP3A4KCNH2ADRB1
SCHEMBL12894526 0.93 CCR1 (0.71) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567500 0.93 CCR1 (0.76) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567517 0.93 CCR1 (0.70) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567625 0.93 CCR1 (0.70) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567101 0.92 CCR1 (0.69) CCR1CYP3A4KCNH2ADRB1
SCHEMBL568675 0.92 CCR1 (0.69) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567612 0.89 CCR1 (0.65) CCR1CYP3A4KCNH2ADRB1
SCHEMBL568650 0.88 CCR1 (0.65) CCR1CYP3A4KCNH2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102227425-A Azaindazole compounds as ccr1 receptor antagonists BOEHRINGER INGELHEIM INT 2011-10-26 CN disclosed
EP-2346868-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-27 EP disclosed
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed