SCHEMBL23019685

SCHEMBL23019685

CC(C)(C)OC(=O)N1CCC(NC(=O)c2ccc(Br)cc2F)C1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 12/20 0.70
FPR3 P25089 2/20 0.51
FPR2 P25090 2/20 0.51
RIPK1 Q13546 1/20 0.50
HDAC4 P56524 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
PARP1 P09874 1/20 0.49
PBK Q96KB5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18124204 1.00 USP30 (0.70) USP30FPR3FPR2RIPK1HDAC4
SCHEMBL29779090 1.00 USP30 (0.70) USP30FPR3FPR2RIPK1HDAC4
SCHEMBL28513485 0.88 USP30 (0.67) USP30RIPK1HDAC4HDAC6PARP1
SCHEMBL18124183 0.88 USP30 (0.67) USP30RIPK1HDAC4HDAC6PARP1
SCHEMBL29778997 0.88 USP30 (0.67) USP30RIPK1HDAC4HDAC6PARP1
SCHEMBL18115999 0.83 USP30 (0.49) USP30
SCHEMBL19990877 0.83 USP30 (0.49) USP30
SCHEMBL3720765 0.82 USP30 (0.65) USP30FPR3FPR2HDAC4HDAC6
SCHEMBL18124184 0.82 USP30 (1.00) USP30FPR3FPR2
SCHEMBL26187387 0.82 USP30 (0.59) USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3943490-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2022-01-26 EP disclosed
EP-3277677-B9 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LTD (GB) 2021-07-14 EP disclosed
EP-3842427-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2021-06-30 EP disclosed
CN-112707893-A 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2021-04-27 CN disclosed
EP-3277677-B1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LTD (GB) 2021-02-24 EP disclosed
CN-107484415-B 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2021-01-29 CN disclosed