SCHEMBL23024976

SCHEMBL23024976

CC(C)(C)OC(=O)Nc1cc(Cl)ncc1C=N

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.40
MAPKAPK2 P49137 2/20 0.38
AAK1 Q2M2I8 2/20 0.37
METAP1 P53582 1/20 0.36
MAP4K4 O95819 1/20 0.36
TRPA1 O75762 1/20 0.36
P2RX3 P56373 2/20 0.36
STK17B O94768 1/20 0.35
STK17A Q9UEE5 1/20 0.35
BRD9 Q9H8M2 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
CYP17A1 P05093 1/20 0.34
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23025134 0.85 MAP4K4 (0.40) ATRMAPKAPK2AAK1METAP1MAP4K4
SCHEMBL21262226 0.82 ATR (0.44) ATRMAPKAPK2AAK1METAP1TRPA1
SCHEMBL9939369 0.81 ATR (0.46) ATRMAPKAPK2AAK1METAP1MAP4K4
SCHEMBL31493121 0.80 ATR (0.42) ATRMAPKAPK2AAK1METAP1TRPA1
SCHEMBL4036319 0.80 MAPKAPK2 (0.43) ATRMAPKAPK2AAK1METAP1MAP4K4
SCHEMBL18369794 0.80 ATR (0.42) ATRMAPKAPK2AAK1METAP1TRPA1
SCHEMBL3344049 0.80 AAK1 (0.45) ATRMAPKAPK2AAK1METAP1TRPA1
SCHEMBL24157078 0.80 ATR (0.42) ATRMAPKAPK2AAK1METAP1TRPA1
SCHEMBL15584205 0.80 ATR (0.42) ATRMAPKAPK2AAK1METAP1MAP4K4
SCHEMBL16879643 0.80 ATR (0.44) ATRMAPKAPK2AAK1METAP1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021032582-A1 PYRAZOLO[4,3-C]PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2021-02-25 WO disclosed