SCHEMBL230383

SCHEMBL230383

Cc1cc(-c2cc(O)ccc2Cl)cc2cnc(Nc3ccc(N4CCN(C(=O)c5ccccn5)CC4)cc3)nc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 16/20 0.54
ABL1 P00519 8/20 0.52
PDGFRB P09619 5/20 0.50
YES1 P07947 3/20 0.50
KDR P35968 3/20 0.50
LCK P06239 2/20 0.45
HCK P08631 1/20 0.45
ALK Q9UM73 1/20 0.44
CCNK O75909 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CCND3 P30281 1/20 0.43
CDK9 P50750 1/20 0.43
CDK6 Q00534 1/20 0.43
EPHB4 P54760 2/20 0.43
NAMPT P43490 1/20 0.43
CIT O14578 1/20 0.43
GAK O14976 1/20 0.43
EPHB6 O15197 1/20 0.43
RIPK2 O43353 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL229295 0.89 SRC (0.60) SRCABL1PDGFRBYES1KDR
SCHEMBL230386 0.88 SRC (0.56) SRCABL1PDGFRBYES1KDR
SCHEMBL231132 0.88 ALK (0.58) SRCABL1PDGFRBYES1KDR
SCHEMBL2579072 0.81 SRC (0.52) SRCABL1PDGFRBYES1KDR
SCHEMBL226225 0.72 SRC (0.55) SRCABL1PDGFRBYES1KDR
SCHEMBL2580732 0.72 SRC (0.55) SRCABL1PDGFRBYES1KDR
SCHEMBL231130 0.71 SRC (0.78) SRCABL1PDGFRBYES1KDR
SCHEMBL4264029 0.70 SRC (1.00) SRCABL1PDGFRBYES1KDR
SCHEMBL230633 0.70 SRC (0.49) SRCABL1PDGFRBYES1KDR
SCHEMBL230632 0.70 SRC (0.49) SRCABL1PDGFRBYES1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8389530-B2 Substituted quinazoline compounds FOVEA PHARMACEUTICALS (FR) 2013-03-05 US claimed
US-20120004210-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS FOVEA PHARMACEUTICALS SA 2012-01-05 US claimed
US-8389530-B2 Substituted quinazoline compounds FOVEA PHARMACEUTICALS (FR) 2013-03-05 US disclosed
US-20120004210-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS FOVEA PHARMACEUTICALS SA 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120004210-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS MAP3K5, MAP3K1, MAP3K2 SRC 1325/4885ABL1 442/4885PDGFRB 1013/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.