SCHEMBL23055258

SCHEMBL23055258

CC(C)Nc1ccn2cccc2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP7 Q93009 1/20 0.35
MAP4K4 O95819 1/20 0.35
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KCNH3 Q9ULD8 1/20 0.33
GAA P10253 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
PTGS1 P23219 2/20 0.32
PTGS2 P35354 2/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32
KDM4E B2RXH2 4/20 0.32
HPGD P15428 2/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11989037 0.81 PTGS1 (0.44) USP7ALDH1A1PTGS1PTGS2KDM4E
SCHEMBL13034797 0.74 PCSK9 (0.47) MAP4K4ALDH1A1MEN1KMT2AGAA
SCHEMBL18238797 0.72 NPC1 (0.35) ALDH1A1PTGS1PTGS2KDM4EHPGD
SCHEMBL24783513 0.70 FLT3 (0.34) MAP4K4ALDH1A1MEN1KMT2AGAA
SCHEMBL12541310 0.69 TDP1 (0.44) ALDH1A1MEN1KMT2AKCNH3GAA
SCHEMBL19153502 0.69 NPC1 (0.37) ALDH1A1KMT2AGAATDP1PTGS1
SCHEMBL11989034 0.67 MAP4K4 (0.34) USP7MAP4K4KCNH3TDP1TRPM8
SCHEMBL15679454 0.64 KDM4E (0.35) ALDH1A1KMT2AGAAPTGS1PTGS2
SCHEMBL26247375 0.64 NPC1 (0.41) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL9217808 0.64 PTGS1 (0.52) ALDH1A1PTGS1PTGS2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021149767-A1 HETEROCYCLIC DERIVATIVE 大日本住友製薬株式会社 2021-07-29 WO disclosed
WO-2021039961-A1 RING-FUSED PYRAZOLE DERIVATIVE 大日本住友製薬株式会社 2021-03-04 WO disclosed