SCHEMBL23062897

SCHEMBL23062897

O=C(OCc1ccccc1)[C@H]1C(F)(F)C12CCNCC2

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
HTR2C P28335 1/20 0.41
TACR1 P25103 1/20 0.41
FABP7 O15540 1/20 0.41
FABP5 Q01469 1/20 0.41
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
ALDH1A1 P00352 3/20 0.40
OPRM1 P35372 1/20 0.39
BACE1 P56817 1/20 0.39
GLA P06280 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
FKBP1A P62942 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23068987 1.00 TSHR (0.41) TSHRHTR2CTACR1FABP7FABP5
Hydrochloric Acid SCHEMBL22615982 0.99 TSHR (0.43) TSHRHTR2CTACR1FABP7FABP5
Hydrochloric Acid SCHEMBL23062893 0.99 TSHR (0.43) TSHRHTR2CTACR1FABP7FABP5
SCHEMBL29573141 0.79 CHRNA7 (0.43) TSHRFKBP1A
SCHEMBL22615959 0.79 CHRNA7 (0.43) TSHRFKBP1A
SCHEMBL28501135 0.79 CHRNA7 (0.43) TSHRFKBP1A
SCHEMBL23068811 0.78 CYP2D6 (0.44) TSHRTACR1ALDH1A1L3MBTL1KMT2A
SCHEMBL23062927 0.78 CYP2D6 (0.44) TSHRTACR1ALDH1A1L3MBTL1KMT2A
Hydrochloric Acid SCHEMBL23062917 0.77 TSHR (0.40) TSHRHTR2CFABP7FABP5DDB1
SCHEMBL22615941 0.76 TACR1 (0.49) TACR1L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3788043-A1 SPIROPIPERIDINE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS Merck Sharp & Dohme Corp. (US) 2021-03-10 EP disclosed