SCHEMBL2306541

SCHEMBL2306541

O=C(O)c1cccc(NC(=O)C(C2CCCCC2)C2(C(O)c3ccc(F)cc3)Nc3cc(F)c(F)cc3N2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.43
HTR2B P41595 1/20 0.42
EPHX2 P34913 1/20 0.41
APEX1 P27695 1/20 0.39
ANO1 Q5XXA6 1/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 1/20 0.37
ACKR3 P25106 1/20 0.37
KCNK3 O14649 2/20 0.36
KCNK9 Q9NPC2 2/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTR1E P28566 1/20 0.35
S1PR3 Q99500 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2310577 0.90 NR1H4 (0.42) NR1H4HTR2BEPHX2NPC1RAB9A
SCHEMBL2310551 0.88 NR1H4 (0.41) NR1H4HTR2BEPHX2APEX1ANO1
SCHEMBL2309892 0.88 NR1H4 (0.44) NR1H4HTR2BNPC1RAB9A
SCHEMBL2305348 0.85 NR1H4 (0.46) NR1H4NPC1RAB9A
SCHEMBL2308785 0.78 NR1H4 (0.40) NR1H4HTR2BEPHX2NPC1RAB9A
SCHEMBL2913040 0.77 TSHR (0.44) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL2308591 0.77 NR1H4 (0.43) NR1H4NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL2306977 0.76 NR1H4 (0.43) NR1H4HTR2BEPHX2NPC1RAB9A
SCHEMBL2305595 0.76 NR1H4 (0.49) NR1H4NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL2304490 0.74 NR1H4 (0.44) NR1H4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350022-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-08-03 EP claimed
WO-2010043513-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-04-22 WO claimed