SCHEMBL23119030

SCHEMBL23119030

CNc1ccc(Nc2nc(Nc3ccc(NC(C)=O)cc3)ncc2[N+](=O)[O-])c(C(=O)c2ccccc2)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.83
MAPT P10636 3/20 0.66
PTK2B Q14289 2/20 0.66
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2C9 P11712 1/20 0.66
CYP2C19 P33261 1/20 0.66
MCL1 Q07820 1/20 0.66
GSK3B P49841 6/20 0.56
GSK3A P49840 5/20 0.56
AURKA O14965 3/20 0.56
PTK2 Q05397 6/20 0.49
MAPK1 P28482 2/20 0.49
CDC7 O00311 1/20 0.49
PLK4 O00444 1/20 0.49
CHEK1 O14757 1/20 0.49
DCLK1 O15075 1/20 0.49
CHUK O15111 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032124 0.91 PLK1 (1.00) PLK1MAPTPTK2BMEN1KMT2A
Hydrochloric Acid SCHEMBL3808883 0.90 PLK1 (0.98) PLK1MAPTPTK2BMEN1KMT2A
SCHEMBL4025594 0.84 PLK1 (0.84) PLK1MAPTPTK2BMEN1KMT2A
Hydrochloric Acid SCHEMBL3810870 0.83 PLK1 (0.82) PLK1MAPTPTK2BMEN1KMT2A
SCHEMBL13866466 0.83 PLK1 (0.81) PLK1MAPTPTK2BMEN1KMT2A
Hydrochloric Acid SCHEMBL3814491 0.82 PLK1 (0.80) PLK1MAPTPTK2BMEN1KMT2A
SCHEMBL5408359 0.81 MAPT (0.86) PLK1MAPTPTK2BMEN1KMT2A
SCHEMBL4031609 0.80 MAPT (0.70) PLK1MAPTPTK2BMEN1KMT2A
Hydrochloric Acid SCHEMBL3814985 0.79 MAPT (0.69) PLK1MAPTPTK2BMEN1KMT2A
SCHEMBL13866473 0.78 PLK1 (0.72) PLK1MAPTPTK2BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021050917-A1 PHOSPHOLIPID ETHER CONJUGATES AS CANCER-TARGETING DRUG VEHICLES CELLECTAR BIOSCIENCES, INC. (US) 2021-03-18 WO disclosed