SCHEMBL23134697

SCHEMBL23134697

COc1cc(-c2cc(C)c(=O)n(C)c2)c(OC)cc1C

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 20/20 0.67
BRD9 Q9H8M2 11/20 0.67
BRD2 P25440 3/20 0.53
BRD7 Q9NPI1 3/20 0.53
BAZ2A Q9UIF9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23121920 0.85 BRD4 (0.62) BRD4BRD9BRD2BRD7
SCHEMBL23134772 0.81 BRD4 (0.51) BRD4BRD9BRD2BRD7
SCHEMBL19869744 0.81 BRD9 (1.00) BRD4BRD9BRD2BRD7
SCHEMBL23134715 0.79 BRD9 (0.49) BRD4BRD9BRD2BRD7
SCHEMBL23134730 0.78 BRD4 (0.67) BRD4BRD9BRD2BRD7
SCHEMBL23134702 0.78 BRD4 (0.65) BRD4BRD9BRD2BRD7
SCHEMBL23134699 0.78 BRD4 (0.68) BRD4BRD9BRD2BRD7
SCHEMBL19869726 0.77 BRD4 (0.65) BRD4BRD9BRD2BRD7
SCHEMBL19869734 0.77 MAPT (0.57) BRD4BRD9BRD2BRD7
SCHEMBL24556425 0.76 BRD4 (0.52) BRD4BRD9BRD2BRD7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021055295-A1 BRD9 BIFUNCTIONAL DEGRADERS AND THEIR METHODS OF USE NOVARTIS AG (CH) 2021-03-25 WO disclosed