SCHEMBL23222858

SCHEMBL23222858

C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@H]3C(CC[C@]12C)[C@@]1(C)CC[C@@H](OC(=O)CC[C@@H](C)[C@H]2CC[C@H]4[C@@H]5[C@@H](O)C[C@@H]6C[C@H](O)CC[C@]6(C)[C@H]5CC[C@]24C)C[C@H]1C[C@@H]3O

nearest known ligand 0.82

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 13/20 0.82
NR1H4 Q96RI1 5/20 0.82
ABCB11 O95342 3/20 0.82
MEN1 O00255 2/20 0.82
KMT2A Q03164 2/20 0.82
SLC10A2 Q12908 2/20 0.82
SLC10A1 Q14973 2/20 0.82
ENPP2 Q13822 2/20 0.82
LMNA P02545 1/20 0.82
CYP2C19 P33261 1/20 0.82
CHRM2 P08172 1/20 0.82
ADRA2A P08913 1/20 0.82
ADRA1A P35348 1/20 0.82
TDP1 Q9NUW8 1/20 0.82
CISD1 Q9NZ45 1/20 0.82
CYP3A4 P08684 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532588 1.00 GPBAR1 (0.82) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL1551522 1.00 GPBAR1 (0.82) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL10717974 1.00 GPBAR1 (0.82) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL13584586 0.97 GPBAR1 (0.77) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL517850 0.95 GPBAR1 (0.74) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL2638871 0.95 GPBAR1 (0.74) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL1287858 0.94 GPBAR1 (0.78) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL15558007 0.92 GPBAR1 (0.70) GPBAR1NR1H4ABCB11MEN1KMT2A
SCHEMBL23231228 0.91 GPBAR1 (0.81) GPBAR1NR1H4ABCB11MEN1KMT2A
Chenodiol SCHEMBL25337643 0.91 GPBAR1 (1.00) GPBAR1NR1H4ABCB11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3804750-A1 CONJUGATE COMPOUNDS FOR PREVENTING AND/OR TREATING HBV AND/OR HDV INFECTIONS, LIVER DISEASES AND FOR TARGETING NTCP Universität Heidelberg (DE) 2021-04-14 EP disclosed