SCHEMBL2323372

SCHEMBL2323372

CN(C(=O)N(c1c(Cl)cccc1Cl)c1c(Cl)cccc1Cl)c1cc(Nc2cccc(C#N)c2)ncn1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LCK P06239 13/20 0.48
CYP3A4 P08684 2/20 0.42
FGFR3 P22607 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2C9 P11712 1/20 0.41
EGFR P00533 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
GRM4 Q14833 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
F9 P00740 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374251 0.84 LCK (0.69) LCKCYP3A4FGFR3CYP2C19CYP2C9
SCHEMBL374267 0.70 LCK (0.76) LCKCYP3A4FGFR3CYP2C19CYP2C9
SCHEMBL374265 0.70 TNNI3K (0.56) EGFRABCG2F9
SCHEMBL374719 0.69 LCK (0.73) LCKCYP3A4FGFR3CYP2C19CYP2C9
SCHEMBL374686 0.67 LCK (0.72) LCKCYP3A4FGFR3CYP2C19CYP2C9
SCHEMBL13855375 0.66 LCK (0.58) LCKCYP3A4FGFR3CYP2C19EGFR
SCHEMBL374147 0.65 LCK (1.00) LCKCYP3A4FGFR3CYP2C19
SCHEMBL374072 0.65 LCK (0.62) LCKCYP3A4FGFR3CYP2C19CYP2C9
SCHEMBL374236 0.65 LCK (0.79) LCKCYP3A4FGFR3CYP2C19
SCHEMBL27320738 0.64 KDM1A (0.48) CYP2C19EGFRABCG2IRAK4F9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761505-B1 PYRIMIDINE UREA DERIVATIVES AS KINASE INHIBITORS NOVARTIS AG (CH) 2011-08-17 EP disclosed