SCHEMBL2324960

SCHEMBL2324960

Nc1nnc(-c2cc(Br)nc(C(F)(F)F)c2)c(-c2ccccc2)n1.Nc1nnc(-c2cc(Cl)nc(C(F)(F)F)c2)c(-c2ccccc2)n1

nearest known ligand 0.69

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.69
ADORA1 P30542 19/20 0.69
ADORA2B P29275 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2329561 0.93 ADORA2A (0.73) ADORA2AADORA1ADORA2B
SCHEMBL2323998 0.93 ADORA2A (0.79) ADORA2AADORA1ADORA2B
SCHEMBL2319984 0.84 ADORA2A (0.82) ADORA2AADORA1ADORA2B
SCHEMBL2322065 0.82 ADORA2A (1.00) ADORA2AADORA1ADORA2B
SCHEMBL2322516 0.81 ADORA2A (0.76) ADORA2AADORA1ADORA2B
SCHEMBL17667882 0.81 ADORA2A (0.52) ADORA2AADORA1ADORA2B
SCHEMBL2321400 0.80 ADORA2A (0.81) ADORA2AADORA1ADORA2B
SCHEMBL2323349 0.79 ADORA2A (0.81) ADORA2AADORA1ADORA2B
SCHEMBL2323578 0.79 ADORA2A (0.75) ADORA2AADORA1ADORA2B
SCHEMBL2327585 0.78 ADORA2A (1.00) ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531492-A1 1,2,4-TRIAZINE-4-AMINE DERIVATIVES Heptares Therapeutics Limited (GB) 2012-12-12 EP claimed
WO-2011095625-A1 1,2,4-TRIAZINE-4-AMINE DERIVATIVES HEPTARES THERAPEUTICS LIMITED (GB) 2011-08-11 WO claimed