SCHEMBL2325347

SCHEMBL2325347

C[N+]1(C)c2ccc(C#Cc3ccc(-c4ccc(Cl)cc4)cn3)cc2CCC1N1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.47
CHRM1 P11229 5/20 0.46
HTR2A P28223 4/20 0.46
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4512906 0.79 MCHR1 (0.50) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4503035 0.73 MCHR1 (0.55) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2323297 0.72 MCHR1 (0.53) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2326974 0.70 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4519018 0.70 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2321880 0.69 MCHR1 (0.62) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5230226 0.68 MCHR1 (0.61) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL13933782 0.68 MCHR1 (0.53) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2324871 0.68 MCHR1 (0.53) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5220840 0.68 MCHR1 (0.57) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed