SCHEMBL23296207

SCHEMBL23296207

CN1CC2CCC(C1)N2Cc1ccc(Nc2ncccn2)nc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.40
JAK2 O60674 3/20 0.39
JAK1 P23458 3/20 0.39
TYK2 P29597 3/20 0.39
CNR2 P34972 6/20 0.39
CCND1 P24385 6/20 0.37
CDK6 Q00534 6/20 0.37
CDK2 P24941 2/20 0.36
CCNT1 O60563 1/20 0.36
CDK4 P11802 1/20 0.36
CCNA2 P20248 1/20 0.36
CCND3 P30281 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36
CCNH P51946 1/20 0.36
CDK1 P06493 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23296212 0.89 CNR2 (0.40) IDH1CNR2
SCHEMBL20744436 0.88 TLR7 (0.40) CNR2CCND1CDK6CDK2CDK4
SCHEMBL23296205 0.83 CDK6 (0.43) IDH1CNR2CCND1CDK6CDK2
SCHEMBL20744900 0.81 CNR2 (0.42) IDH1CNR2CCND1CDK6CDK2
SCHEMBL29686224 0.78 CCND1 (0.43) CNR2CCND1CDK6CDK2CDK4
SCHEMBL20744557 0.77 CCND1 (0.54) CCND1CDK6CDK2CDK4CCNA2
SCHEMBL20744015 0.75 CCND1 (0.42) CNR2CCND1CDK6CDK2CCNT1
SCHEMBL29615707 0.73 CHRM2 (0.49)
SCHEMBL20744508 0.73 CCND1 (0.46) CCND1CDK6CDK2CDK4CCNA2
SCHEMBL29615744 0.73 CYP11B1 (0.40) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11351170-B2 Substituted pyrimidines as CDK4/6 inhibitors BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2022-06-07 US disclosed
US-20210128555-A1 CDK4/6 INHIBITORS AND USE THEREOF BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2021-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11351170-B2 Substituted pyrimidines as CDK4/6 inhibitors CDK4, CDK6, CDK2 IDH1 190/4885JAK2 89/4885JAK1 106/4885
US-20210128555-A1 CDK4/6 INHIBITORS AND USE THEREOF CDK4, CDK6, CDK1 IDH1 281/4885JAK2 71/4885JAK1 84/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.