SCHEMBL2330973

SCHEMBL2330973

COCCN1C(=O)c2ccccc2C(C(=O)Nc2cccc(OC)c2)C1c1c(F)cccc1F.COCCN1C(=O)c2ccccc2C(C(=O)Nc2cccc(OC)c2)C1c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.67
CYP2C19 P33261 1/20 0.67
ALDH1A1 P00352 4/20 0.64
KDM4E B2RXH2 3/20 0.64
MAPT P10636 3/20 0.64
HTT P42858 1/20 0.64
GAA P10253 2/20 0.63
TSHR P16473 2/20 0.60
NPSR1 Q6W5P4 3/20 0.58
L3MBTL1 Q9Y468 1/20 0.53
HSD17B10 Q99714 1/20 0.51
NPC1 O15118 2/20 0.49
FFAR1 O14842 1/20 0.47
TP53 P04637 1/20 0.45
MDM2 Q00987 1/20 0.45
CYP3A4 P08684 1/20 0.43
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2333798 0.95 GAA (0.61) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2337037 0.95 CYP2C9 (0.73) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2330237 0.89 GAA (0.62) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2335360 0.89 GAA (0.69) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2334762 0.89 CYP2C9 (0.64) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2336094 0.88 GAA (0.67) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2334971 0.87 GAA (0.66) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2336153 0.84 GAA (0.64) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2331052 0.83 GAA (0.61) CYP2C9CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL2339500 0.83 GAA (0.70) CYP2C9CYP2C19ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358682-A2 ISOQUINOLONE DERIVATIVES AS INHIBITORS OF PLAVIVIRUS REPLICATION Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2011-08-24 EP disclosed