SCHEMBL23339883

SCHEMBL23339883

CCCNc1ncnc2cc(Cl)ccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.60
PPARG P37231 1/20 0.60
NR2E3 Q9Y5X4 1/20 0.60
NCOR2 Q9Y618 1/20 0.60
HTT P42858 6/20 0.59
SMN1; SMN2 Q16637 4/20 0.59
LMNA P02545 2/20 0.59
CCNC P24863 1/20 0.58
CDK8 P49336 1/20 0.58
KDM4E B2RXH2 2/20 0.58
ALDH1A1 P00352 2/20 0.58
HPGD P15428 1/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
NPC1 O15118 1/20 0.56
STAT1 P42224 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
MAPK1 P28482 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31089964 0.91 SMN1; SMN2 (0.58) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL11846406 0.91 KDM4E (0.63) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL15923148 0.89 SMN1; SMN2 (0.67) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL31197395 0.89 SMN1; SMN2 (0.67) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL15924449 0.89 SMN1; SMN2 (0.67) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL11855329 0.86 HDAC1 (0.60) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL11857739 0.86 HDAC1 (0.60) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL11849897 0.86 HDAC1 (0.60) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL18290260 0.84 RXFP1 (0.56) RXFP1PPARGNR2E3NCOR2HTT
SCHEMBL24652841 0.84 RXFP1 (0.56) RXFP1PPARGNR2E3NCOR2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022250971-A1 SMALL MOLECULE INHIBITORS OF AUTOPHAGY AND HISTONE DEACTYLASES AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2022-12-01 WO disclosed
WO-2021087077-A1 SMALL MOLECULE INHIBITORS OF AUTOPHAGY AND HISTONE DEACTYLASES AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2021-05-06 WO disclosed