SCHEMBL23368182

SCHEMBL23368182

COc1cc2ncnc(Nc3ccc(Oc4cccc(-c5nnc(C(C)C)o5)c4)cc3F)c2cc1N

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.47
FLT1 P17948 6/20 0.47
KDR P35968 10/20 0.46
FGFR1 P11362 3/20 0.46
RET P07949 5/20 0.45
KIF5B P33176 5/20 0.45
EPHB2 P29323 2/20 0.45
FLT4 P35916 2/20 0.45
RIPK2 O43353 1/20 0.41
CCNT1 O60563 1/20 0.41
GSK3B P49841 1/20 0.41
CDK9 P50750 1/20 0.41
DYRK1A Q13627 1/20 0.41
ERBB4 Q15303 1/20 0.40
MAPK14 Q16539 1/20 0.40
RAF1 P04049 1/20 0.39
BRAF P15056 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21616332 0.90 EGFR (0.48) EGFRFLT1KDRFGFR1RET
SCHEMBL30203115 0.90 EGFR (0.48) EGFRFLT1KDRFGFR1RET
SCHEMBL23368026 0.88 EGFR (0.48) EGFRFLT1KDRFGFR1RET
SCHEMBL23355476 0.88 EGFR (0.47) EGFRFLT1KDRFGFR1RET
SCHEMBL23355432 0.82 EGFR (0.47) EGFRFLT1KDRFGFR1RET
SCHEMBL23355452 0.82 EGFR (0.47) EGFRFLT1KDRFGFR1RET
SCHEMBL21616356 0.82 EGFR (0.55) EGFRKDRERBB4
SCHEMBL23368220 0.81 EGFR (0.49) EGFRFLT1KDRFGFR1RET
SCHEMBL24037410 0.81 KDR (0.52) EGFRFLT1KDRFGFR1RET
SCHEMBL23368122 0.79 EGFR (0.48) EGFRFLT1KDRFGFR1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230025510-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVES DAIICHI SANKYO COMPANY, LIMITED (JP) 2023-01-26 US disclosed
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230025510-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVES ERBB2, EGFR, ERBB3 EGFR 2/4885FLT1 119/4885KDR 20/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.