SCHEMBL2344949

SCHEMBL2344949

CC(C)NC(=O)Oc1c[nH]c2ncc(-c3cccc(S(C)(=O)=O)c3)nc12

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.46
CYP2C9 P11712 1/20 0.46
JAK3 P52333 6/20 0.44
ATR Q13535 3/20 0.43
PRKDC P78527 1/20 0.43
ATM Q13315 1/20 0.43
CAMKK2 Q96RR4 2/20 0.43
BTK Q06187 1/20 0.41
ITK Q08881 1/20 0.41
KCNH2 Q12809 2/20 0.40
PLK4 O00444 1/20 0.40
MAPK1 P28482 1/20 0.39
JAK2 O60674 4/20 0.39
JAK1 P23458 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2276326 0.85 SYK (0.61) SYKCYP2C9JAK3ATRPRKDC
SCHEMBL2344042 0.84 SYK (0.52) SYKCYP2C9JAK3ATRPRKDC
SCHEMBL2349746 0.83 SYK (0.49) SYKCYP2C9JAK3MAPK1JAK2
SCHEMBL2342514 0.83 JAK3 (0.49) SYKCYP2C9JAK3ATRBTK
SCHEMBL2347616 0.83 SYK (0.46) SYKCYP2C9JAK3MAPK1JAK2
SCHEMBL2342554 0.80 ATR (0.46) SYKCYP2C9JAK3ATRPLK4
SCHEMBL2339099 0.80 SYK (0.62) SYKCYP2C9JAK3ATMMAPK1
SCHEMBL2341691 0.77 SYK (0.43) SYKCYP2C9JAK3JAK2JAK1
SCHEMBL2344083 0.76 SYK (0.49) SYKCYP2C9JAK3ATRMAPK1
SCHEMBL2346514 0.76 SYK (0.49) SYKCYP2C9JAK3MAPK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245033-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2011-08-31 EP claimed