SCHEMBL23478

SCHEMBL23478

COc1cc(CCN)c(OC)cc1Br

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 13/20 1.00
TAAR1 Q96RJ0 6/20 1.00
HTR2C P28335 4/20 1.00
HTR2B P41595 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29351348 1.00 HTR2A (1.00) HTR2ATAAR1HTR2CHTR2B
SCHEMBL5809547 1.00 HTR2A (1.00) HTR2ATAAR1HTR2CHTR2B
Hydrochloric Acid SCHEMBL22614747 0.98 HTR2A (0.96) HTR2ATAAR1HTR2CHTR2B
Methane SCHEMBL20703126 0.98 HTR2A (0.96) HTR2ATAAR1HTR2CHTR2B
Hydrochloric Acid SCHEMBL25285317 0.98 HTR2A (0.96) HTR2ATAAR1HTR2CHTR2B
SCHEMBL31285026 0.92 HTR2A (0.84) HTR2ATAAR1HTR2CHTR2B
SCHEMBL31284837 0.92 HTR2A (0.84) HTR2ATAAR1HTR2CHTR2B
Acetic Acid SCHEMBL31176574 0.90 HTR2A (0.81) HTR2ATAAR1HTR2C
Hydrochloric Acid SCHEMBL30284705 0.90 HTR2A (0.81) HTR2ATAAR1HTR2CHTR2B
Hydrochloric Acid SCHEMBL30284868 0.90 HTR2A (0.81) HTR2ATAAR1HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 32724 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4728531-A1 BIOADAPTIVE THERAPEUTIC ENVIRONMENTS Therapod LLC (US) 2026-04-22 EP claimed
EP-4358962-B1 TREATMENT FOR AUTOIMMUNE DISEASES COMPRISING NALTREXONE OR A METABOLITE OR ANALOG THEREOF, A CANNABINOID AND A 5-HT RECEPTOR AGONIST LDN PHARMA LTD (GB) 2026-02-04 EP claimed
US-12514883-B2 Compositions and methods for modulating lipid and steroid metabolism THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-01-06 US claimed
US-20250360150-A1 METHODS OF USING NEUROPLASTIC AGENTS AND TERRAFORMING MARS BRANNOCK METCALF MOLLY CAROLINE (US) 2025-11-27 US claimed
US-12465275-B2 Molecularly-initiated, experientially-delivered treatments and systems for practicing same THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-11-11 US claimed
EP-4633638-A1 TREATMENT OF PSYCHOLOGICAL FACTORS AFFECTING OTHER MEDICAL CONDITIONS (PFAOMC) Luminous Mind Inc. (US) 2025-10-22 EP claimed
EP-4615585-A1 METHODS OF USING TRAZODONE TO REVERSE THE EFFECTS OF 5-HT2A RECEPTOR AGONISTS Gilgamesh Pharmaceuticals, Inc. (US) 2025-09-17 EP claimed
US-20250281481-A1 NALTREXONE FOR BOOSTING THE THERAPEUTIC UTILTY OF 5-HT RECEPTOR AGONISTS LDN Pharma Limited (GB) 2025-09-11 US claimed
EP-4547250-A1 METHODS AND COMPOSITIONS RELATING TO CONTROLLING PSYCHEDELIC EFFECTS WITH SEROTONIN RECEPTOR MODULATORS Terran Biosciences Inc. (US) 2025-05-07 EP claimed
WO-2025030181-A1 CRYSTALLINE POLYMORPHS OF 4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE (2C-B) ARCADIA MEDICINE, INC. (US) 2025-02-06 WO claimed
EP-0080616-A1 Gas borne particle filtering method Long, James (US) 1983-06-08 EP claimed
EP-0071359-A1 Methods and apparatus for molten metal fume supression USS ENGINEERS AND CONSULTANTS, INC. (US) 1983-02-09 EP claimed
EP-0062667-A1 IMPROVED SYSTEM FOR INTERRUPT ARBITRATION. DIGITAL EQUIPMENT CORP (US) 1982-10-20 EP claimed
US-4339816-A Conferencing apparatus and methods for a frequency division multiplex communications system INTERNATIONAL TELEPHONE AND TELEGRAPH CORPORATION (US) 1982-07-13 US claimed
WO-1982001430-A1 IMPROVED SYSTEM FOR INTERRUPT ARBITRATION DIGITAL EQUIPMENT CORP (US) 1982-04-29 WO claimed
US-4232366-A Bus for a data processing system with overlapped sequences DIGITAL EQUIPMENT CORPORATION (US) 1980-11-04 US claimed
US-4229791-A Distributed arbitration circuitry for data processing system DIGITAL EQUIPMENT CORPORATION (US) 1980-10-21 US claimed
US-4135894-A Air filtration apparatus and method of operation thereof ANDERSEN 2000, INC. (US) 1979-01-23 US claimed
US-4038775-A Doll body with magnet and pole pieces and detachable appendages TAKARA CO, LTD. (JA) 1977-08-02 US claimed
US-3993224-A Spout for two-component resin dispenser AEROSOL INVESTMENTS, LTD. (US) 1976-11-23 US claimed