SCHEMBL23501892

SCHEMBL23501892

CCCC(=O)NC(Cc1c[nH]c2ccc(O)cc12)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.60
NFKB1 P19838 3/20 0.60
BLM P54132 2/20 0.60
HTR1A P08908 2/20 0.60
HTR2A P28223 2/20 0.60
HTR2C P28335 2/20 0.60
HTR2B P41595 2/20 0.60
KMT2A Q03164 2/20 0.60
ALDH1A1 P00352 2/20 0.60
LMNA P02545 2/20 0.60
TSHR P16473 2/20 0.60
PMP22 Q01453 2/20 0.60
KDM4E B2RXH2 1/20 0.60
CYP3A4 P08684 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
MAPT P10636 1/20 0.60
ALOX15 P16050 1/20 0.60
SLC6A4 P31645 1/20 0.60
HTR7 P34969 1/20 0.60
MTOR P42345 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23501891 1.00 NPSR1 (0.60) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL23501894 0.93 TRPV1 (0.64) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL23501893 0.93 TRPV1 (0.64) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL27964771 0.91 NPSR1 (0.60) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL11486816 0.89 NPSR1 (0.59) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL11486815 0.89 NPSR1 (0.59) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL23501871 0.89 GAA (0.58) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL23501868 0.89 GAA (0.58) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL23501915 0.88 KMT2A (0.62) NPSR1NFKB1BLMHTR1AHTR2A
SCHEMBL23501914 0.88 KMT2A (0.62) NPSR1NFKB1BLMHTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021118318-A2 NOVEL INDOLE DERIVATIVE AND USE THEREOF 주식회사 메타센테라퓨틱스 2021-06-17 WO disclosed
CN-103804270-B 5-(4-amidino benzyloxy) tryptophan derivative, its method for making and application 中国药科大学 2016-06-22 CN disclosed
CN-103755686-B The piperidyl with platelet aggregation inhibitory activity replaces 5-hydroxyryptophan derivative CHINA PHARMACEUTICAL UNIVERSITY (CN) 2016-05-11 CN disclosed
CN-103804270-A 5-(4-amidinobenzyloxy) tryptophan derivatives and preparation method and application thereof UNIV CHINA PHARMA 2014-05-21 CN disclosed
CN-103755686-A Piperidyl substituted 5-hydroxytryptophane derivatives with anti-platelet aggregation activity UNIV CHINA PHARMA 2014-04-30 CN disclosed