SCHEMBL2357708

SCHEMBL2357708

CC(C)(C)Nc1ncccc1-c1nnnn1-c1ccc(N2CCN(C(=O)O)CC2)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
KCNN4 O15554 5/20 0.35
TRPV1 Q8NER1 2/20 0.35
NPY2R P49146 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GRM5 P41594 1/20 0.33
GRM1 Q13255 1/20 0.33
HSD11B1 P28845 1/20 0.32
AKT1 P31749 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2359384 0.90 AKT1 (0.42) GAAGRM5GRM1AKT1LMNA
SCHEMBL1425424 0.81 KCNN4 (0.44) KCNN4ALDH1A1
SCHEMBL1425298 0.80 KCNN4 (0.46) KCNN4ALDH1A1
SCHEMBL1425971 0.78 KCNN4 (0.38) KCNN4ALDH1A1
SCHEMBL2358883 0.78 KCNN4 (0.46) KCNN4ALDH1A1
SCHEMBL983904 0.77 KCNN4 (0.50) KCNN4
SCHEMBL2359723 0.76 BACE1 (0.38) LMNASMN1; SMN2
SCHEMBL987754 0.76 KCNN4 (0.47) KCNN4ALDH1A1
SCHEMBL2359902 0.72 RET (0.49)
SCHEMBL982800 0.72 KCNN4 (0.46) KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350045-A1 C-MET PROTEIN KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2011-08-03 EP disclosed
WO-2010048131-A1 C-MET PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-04-29 WO disclosed