SCHEMBL2359244

SCHEMBL2359244

Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1NC(=O)c1csc2c(SS(C)(=O)=O)ncnc12

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 5/20 0.56
MAPK14 Q16539 4/20 0.56
KIT P10721 3/20 0.56
SRC P12931 2/20 0.56
RAF1 P04049 2/20 0.53
CSF1R P07333 1/20 0.52
POLB P06746 4/20 0.52
MAPT P10636 3/20 0.52
KDM4E B2RXH2 2/20 0.52
HTT P42858 1/20 0.51
ATM Q13315 1/20 0.51
KDR P35968 3/20 0.51
APEX1 P27695 1/20 0.49
BRAF P15056 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14717890 0.91 LCK (0.59) LCKMAPK14KITSRCRAF1
SCHEMBL2314975 0.86 RAF1 (0.63) LCKMAPK14KITSRCRAF1
SCHEMBL12432525 0.86 LCK (0.61) LCKMAPK14KITSRCRAF1
SCHEMBL2359154 0.84 LCK (0.58) LCKMAPK14KITSRCRAF1
SCHEMBL12432594 0.83 LCK (0.57) LCKMAPK14KITSRCRAF1
SCHEMBL2314225 0.82 LCK (0.56) LCKMAPK14KITSRCRAF1
SCHEMBL2315495 0.82 SRC (0.57) LCKMAPK14KITSRCRAF1
SCHEMBL2314639 0.81 MAPK14 (0.57) LCKMAPK14KITSRCRAF1
SCHEMBL12432595 0.81 BRAF (0.57) LCKMAPK14KITSRCRAF1
SCHEMBL12433876 0.80 BRAF (0.60) LCKMAPK14KITSRCRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed