SCHEMBL2359271

SCHEMBL2359271

CS(=O)(=O)c1cc(-c2nc3cccc(C(F)(F)F)c3nc2N)ccc1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 11/20 0.52
NR1H3 Q13133 7/20 0.52
PTPN1 P18031 1/20 0.39
ALOX5AP P20292 3/20 0.38
FEN1 P39748 3/20 0.38
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2318560 0.88 NR1H2 (0.66) NR1H2NR1H3
SCHEMBL2359274 0.88 NR1H2 (0.51) NR1H2NR1H3PTPN1ALOX5APFEN1
SCHEMBL2319295 0.82 NR1H2 (0.69) NR1H2NR1H3
SCHEMBL2319004 0.81 NR1H2 (0.71) NR1H2NR1H3
SCHEMBL2359416 0.80 NR1H2 (0.48) NR1H2NR1H3ALOX5APFEN1
SCHEMBL2323639 0.80 NR1H2 (0.62) NR1H2NR1H3
SCHEMBL2358913 0.80 NR1H2 (0.45) NR1H2NR1H3ALOX5APFEN1
SCHEMBL3490930 0.80 NR1H2 (0.78) NR1H2NR1H3
SCHEMBL2323837 0.79 NR1H2 (0.65) NR1H2NR1H3
SCHEMBL2358272 0.79 NR1H2 (0.40) NR1H2NR1H3ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2352725-A1 QUINOXALINE-BASED LXR MODULATORS Wyeth LLC (US) 2011-08-10 EP disclosed
WO-2010054229-A1 QUINOXALINE-BASED LXR MODULATORS WYETH LLC (US) 2010-05-14 WO disclosed