SCHEMBL23600433

SCHEMBL23600433

O=C1NCO/C1=C\c1c[nH]c2ncccc12

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.55
CHEK1 O14757 2/20 0.53
HASPIN Q8TF76 4/20 0.53
CDC7 O00311 8/20 0.52
CCNT1 O60563 2/20 0.51
CDK9 P50750 2/20 0.51
PIM1 P11309 2/20 0.45
PIM2 Q9P1W9 2/20 0.45
PIM3 Q86V86 1/20 0.43
GSK3B P49841 1/20 0.43
AXL P30530 1/20 0.41
CHEK2 O96017 1/20 0.40
CDK1 P06493 1/20 0.40
SRC P12931 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23600199 0.79 CHEK1 (0.56) KMT2ACHEK1HASPINCDC7CCNT1
SCHEMBL23578828 0.76 CHEK1 (0.56) KMT2ACHEK1HASPINCCNT1CDK9
SCHEMBL23578825 0.76 CHEK1 (0.56) KMT2ACHEK1HASPINCCNT1CDK9
SCHEMBL1714207 0.76 KMT2A (0.57) KMT2ACHEK1HASPINCDC7CCNT1
SCHEMBL1714205 0.76 KMT2A (0.57) KMT2ACHEK1HASPINCDC7CCNT1
SCHEMBL23582994 0.74 PIM1 (0.54) KMT2ACHEK1HASPINCCNT1CDK9
SCHEMBL4959425 0.74 PIM1 (0.54) KMT2ACHEK1HASPINCCNT1CDK9
SCHEMBL4959430 0.74 PIM1 (0.54) KMT2ACHEK1HASPINCCNT1CDK9
SCHEMBL12506274 0.74 CHEK1 (0.54) KMT2ACHEK1HASPINCDC7CCNT1
SCHEMBL23600236 0.74 HASPIN (0.54) KMT2ACHEK1HASPINCDC7CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021133037-A1 PYRROLIDINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING BETA-AMYLOID OR TAU PROTEIN-ASSOCIATED DISEASES CONTAINING SAME 연세대학교 산학협력단 2021-07-01 WO disclosed