SCHEMBL2361748

SCHEMBL2361748

O=C(N[C]1CCCCCCC1)Nc1n[nH]c2c(F)c(Cl)c(-c3ccccc3)cc12.[CH2].[CH2]

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.63
CDK2 P24941 3/20 0.63
CDK1 P06493 2/20 0.63
GSK3A P49840 4/20 0.38
MAPK1 P28482 9/20 0.37
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2339971 0.86 GSK3B (0.70) GSK3BCDK2CDK1MAPK1
SCHEMBL2361722 0.83 GSK3B (0.62) GSK3BCDK2CDK1GSK3A
SCHEMBL4393025 0.83 GSK3B (0.67) GSK3BCDK2CDK1GSK3AMAPK1
SCHEMBL2335118 0.83 GSK3B (0.67) GSK3BCDK2CDK1MAPK1CYP1A2
SCHEMBL4384920 0.83 GSK3B (0.67) GSK3BCDK2CDK1
SCHEMBL2360845 0.81 GSK3B (0.67) GSK3BCDK2CDK1MAPK1CYP1A2
SCHEMBL2331113 0.81 GSK3B (0.73) GSK3BCDK2CDK1GSK3AMAPK1
SCHEMBL4380218 0.81 GSK3B (0.70) GSK3BCDK2CDK1MAPK1
SCHEMBL4380398 0.80 GSK3B (0.62) GSK3BCDK2CDK1
SCHEMBL4379033 0.80 GSK3B (0.62) GSK3BCDK2CDK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1572200-B1 AMINOINDAZOLE DERIVATIVES AND USE THEREOF AS KINASE INHIBITORS AVENTIS PHARMA SA (FR) 2011-08-17 EP claimed