SCHEMBL2362402

SCHEMBL2362402

C#CCC1(c2ccc3sccc3c2)C=CN=C1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
KCNH2 Q12809 1/20 0.33
DYRK1A Q13627 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361887 0.79 SLC6A2 (0.53) CYP2A6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL984013 0.66 SLC6A2 (0.65) CYP2A6SLC6A2SLC6A4SLC6A3KCNH2
Hydrochloric Acid SCHEMBL984677 0.65 SLC6A2 (0.64) CYP2A6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL984326 0.61 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL9431320 0.59 CYP2A6 (0.46) CYP2A6SLC6A2SLC6A4SLC6A3DYRK1A
SCHEMBL317858 0.56 CYP2A6 (0.50) CYP2A6DYRK1A
SCHEMBL8342108 0.56 CYP2A6 (0.50) CYP2A6DYRK1A
SCHEMBL1426726 0.54 SLC6A4 (0.40) CYP2A6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL164774 0.54 CYP2A6 (0.50) CYP2A6DYRK1A
SCHEMBL17010916 0.54 CYP2A6 (0.52) CYP2A6DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257545-B1 PYRROLIDINYL DERIVATIVES AND USES THEREOF HOFFMANN LA ROCHE (CH) 2011-08-31 EP disclosed