SCHEMBL23628974

SCHEMBL23628974

COC(=O)c1ccc2nc(NC(=O)c3cc(Br)c(Br)[nH]3)sc2c1.O=C(O)c1ccc2nc(NC(=O)c3cc(Br)c(Br)[nH]3)sc2c1

nearest known ligand 0.86

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.62
HTT P42858 1/20 0.58
PIK3CA P42336 1/20 0.58
PIK3CB P42338 1/20 0.58
PIK3CG P48736 1/20 0.58
PI4KB Q9UBF8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23628902 0.96 SCD (0.64) SCDHTTPIK3CAPIK3CBPIK3CG
SCHEMBL23628918 0.93 HSD17B10 (0.56)
SCHEMBL23628978 0.84 SMN1; SMN2 (0.52)
SCHEMBL23628888 0.80 SCD (0.64) SCDHTTPIK3CAPIK3CBPIK3CG
SCHEMBL23628994 0.80
SCHEMBL23629049 0.79 MEN1 (0.42) SCDHTT
SCHEMBL29947440 0.78 HSD17B10 (0.61) SCDHTT
SCHEMBL14807016 0.78 SCD (0.77) SCDHTTPIK3CAPIK3CBPIK3CG
SCHEMBL24729463 0.78 HSD17B10 (0.61) SCDHTT
SCHEMBL24729491 0.77 SCD (0.63) SCDHTTPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3847172-A1 NEW CLASS OF DNA GYRASE AND/OR TOPOISOMERASE IV INHIBITORS WITH ACTIVITY AGAINST GRAM-POSITIVE AND GRAM-NEGATIVE BACTERIA Univerza v Ljubljani (SI) 2021-07-14 EP disclosed