SCHEMBL23637017

SCHEMBL23637017

Cc1c(Nc2ccc(OC(F)(F)F)cc2)ncnc1-c1ccc(N=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 15/20 0.48
BCR P11274 15/20 0.48
TTBK1 Q5TCY1 1/20 0.46
TTBK2 Q6IQ55 1/20 0.46
DHODH Q02127 2/20 0.42
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18696393 0.87 ABL1 (0.53) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL3402884 0.85 ABL1 (0.51) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL17487035 0.84 ABL1 (0.50) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL12943130 0.84 ABL1 (0.57) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL3401859 0.83 ABL1 (0.52) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL3397117 0.83 DHODH (0.50) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL18696394 0.83 ABL1 (0.47) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL3397912 0.83 ABL1 (0.61) ABL1BCRTTBK1TTBK2
SCHEMBL18696249 0.82 ABL1 (0.48) ABL1BCRTTBK1TTBK2DHODH
SCHEMBL18696183 0.82 ABL1 (0.51) ABL1BCRTTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3536687-B1 SMALL MOLECULE MYRISTATE INHIBITORS OF BCR-ABL AND METHODS OF USE DANA FARBER CANCER INST INC (US) 2021-07-14 EP disclosed