SCHEMBL23640504

SCHEMBL23640504

Cc1ccc2c(ccc3onc([C@H]4CCC(=O)NC4=O)c32)c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 17/20 0.42
CRBN Q96SW2 17/20 0.42
SIRT1 Q96EB6 1/20 0.38
IDO1 P14902 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23640500 1.00 DDB1 (0.42) DDB1CRBNSIRT1IDO1SIRT2
SCHEMBL24938749 0.92 DDB1 (0.45) DDB1CRBNIDO1
SCHEMBL24303027 0.87 DDB1 (0.42) DDB1CRBN
SCHEMBL24303033 0.87 DDB1 (0.42) DDB1CRBN
SCHEMBL23639961 0.87 DDB1 (0.52) DDB1CRBN
SCHEMBL23640324 0.87 IDO1 (0.44) DDB1CRBNIDO1
SCHEMBL24303034 0.87 CRBN (0.41) DDB1CRBN
SCHEMBL23639962 0.87 DDB1 (0.52) DDB1CRBN
SCHEMBL23640481 0.87 DDB1 (0.41) DDB1CRBNIDO1
SCHEMBL23640482 0.87 DDB1 (0.41) DDB1CRBNIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3848367-A1 TRICYCLIC COMPOUNDS ACTING ON CRBN PROTEINS Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2021-07-14 EP disclosed