SCHEMBL23670929

SCHEMBL23670929

COC(=O)c1ccc2c(c1)NCC1(CCc3cc(Cl)ccc31)CO2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 14/20 0.45
BCL2L11 O43521 4/20 0.39
ALOX5 P09917 1/20 0.39
RARB P10826 1/20 0.38
RARG P13631 1/20 0.38
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23670931 1.00 MCL1 (0.45) MCL1BCL2L11ALOX5RARBRARG
SCHEMBL17542374 0.94 MCL1 (0.47) MCL1BCL2L11
SCHEMBL29414598 0.94 MCL1 (0.47) MCL1BCL2L11
SCHEMBL17542372 0.94 MCL1 (0.47) MCL1BCL2L11
SCHEMBL23669895 0.90 MCL1 (0.43) MCL1BCL2L11
SCHEMBL23669893 0.90 MCL1 (0.43) MCL1BCL2L11
SCHEMBL19284790 0.90 MCL1 (0.43) MCL1BCL2L11
SCHEMBL29553495 0.90 MCL1 (0.43) MCL1BCL2L11
SCHEMBL29553828 0.90 MCL1 (0.43) MCL1BCL2L11
SCHEMBL19285255 0.88 MCL1 (0.56) MCL1BCL2L11KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12091425-B2 Compounds that inhibit MCL-1 protein AMGEN INC. (US) 2024-09-17 US disclosed
US-20230052348-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN AMGEN INC. (US) 2023-02-16 US disclosed
US-11306107-B2 Compounds that inhibit MCL-1 protein AMGEN INC. (US) 2022-04-19 US disclosed
US-20210230189-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN AMGEN INC. (US) 2021-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210230189-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN MCL1, BCL9, BCL2L1 MCL1 1/4885BCL2L11 7/4885ALOX5 3930/4885
US-11306107-B2 Compounds that inhibit MCL-1 protein MCL1, BCL9, BCL2L1 MCL1 1/4885BCL2L11 7/4885ALOX5 3930/4885
US-20230052348-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN MCL1, BCL9, BCL2L1 MCL1 1/4885BCL2L11 7/4885ALOX5 3930/4885
US-12091425-B2 Compounds that inhibit MCL-1 protein MCL1, BCL9, BCL2L1 MCL1 1/4885BCL2L11 7/4885ALOX5 3930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.