SCHEMBL2369023

SCHEMBL2369023

CCC1(C)CNCCc2cc(OC)c(I)cc21

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 13/20 0.48
HTR2C P28335 13/20 0.48
HTR2B P41595 11/20 0.48
ALDH1A1 P00352 1/20 0.34
DRD1 P21728 1/20 0.32
DRD5 P21918 1/20 0.32
MAOA P21397 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2365641 0.73 HTR2A (0.43) HTR2AHTR2CHTR2BDRD1DRD5
SCHEMBL21661793 0.69 HTR2A (0.59) HTR2AHTR2CHTR2B
SCHEMBL1105042 0.67 HTR2C (0.72) HTR2AHTR2CHTR2BDRD1DRD5
SCHEMBL1095157 0.67 HTR2C (0.72) HTR2AHTR2CHTR2BDRD1DRD5
SCHEMBL1095159 0.67 HTR2C (0.72) HTR2AHTR2CHTR2BDRD1DRD5
SCHEMBL22609757 0.66 HTR2C (0.60) HTR2AHTR2CHTR2BALDH1A1DRD1
SCHEMBL1095292 0.65 HTR2C (1.00) HTR2AHTR2CHTR2B
SCHEMBL1097026 0.65 HTR2C (1.00) HTR2AHTR2CHTR2B
SCHEMBL1097029 0.65 HTR2C (1.00) HTR2AHTR2CHTR2B
SCHEMBL3162737 0.64 HTR2A (0.74) HTR2AHTR2CHTR2BMAOATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2363394-A1 8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine, its salts, solvates or hydrates and its use for the treatment of CNS disorders Arena Pharmaceuticals, Inc. (US) 2011-09-07 EP disclosed