SCHEMBL2369966

SCHEMBL2369966

CCOc1ccc(Cc2cc(C[C@@H]3NC[C@@H](O)[C@H](O)[C@H]3O)ccc2Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC5A2 P31639 18/20 0.51
SLC5A1 P13866 10/20 0.50
ADRA2A P08913 1/20 0.48
SLC5A11 Q8WWX8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16457243 0.83 SLC5A2 (0.59) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL16457244 0.83 SLC5A2 (0.59) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL1039664 0.83 SLC5A2 (0.59) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL2370373 0.78 SLC5A2 (0.49) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL25511558 0.74 SLC5A2 (0.58) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL11313959 0.73 SLC5A2 (0.55) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL28970412 0.73 SLC5A2 (0.74) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL28852291 0.73 SLC5A2 (0.74) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL28970411 0.73 SLC5A2 (0.74) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL1666220 0.73 SLC5A2 (0.72) SLC5A2SLC5A1ADRA2ASLC5A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2661256-A1 COMPOSITIONS COMPRISING AND METHODS OF USING INHIBITORS OF SODIUM-GLUCOSE COTRANSPORTERS 1 AND 2 Lexicon Pharmaceuticals, Inc. (US) 2013-11-13 EP disclosed
EP-2542236-A1 6 -BENZYLPHENYL- 2 - SULFURTERAHYDROPYRAN-3, 4, 5 -TRIOL DERIVATIVES AS INHIBITORS OF SODIUM -GLUCOSE COTRANS PORTERS 1 AND 2 FOR USE IN DIABETIC PATIENTS Lexicon Pharmaceuticals, Inc. (US) 2013-01-09 EP disclosed
WO-2012094293-A1 COMPOSITIONS COMPRISING AND METHODS OF USING INHIBITORS OF SODIUM-GLUCOSE COTRANSPORTERS 1 AND 2 LEXICON PHARMACEUTICALS, INC. (US) 2012-07-12 WO disclosed
WO-2011109333-A1 6 -BENZYLPHENYL- 2 - SULFURTERAHYDROPYRAN-3, 4, 5 -TRIOL DERIVATIVES AS INHIBITORS OF SODIUM -GLUCOSE COTRANS PORTERS 1 AND 2 FOR USE IN DIABETIC PATIENTS LEXICON PHARMACEUTICALS, INC. (US) 2011-09-09 WO disclosed
EP-2089361-A2 INHIBITORS OF SODIUM GLUCOSE CO-TRANSPORTER 2 AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2009-08-19 EP disclosed
WO-2008109591-A1 PHLORIZIN ANALOGS AS INHIBITORS OF SODIUM GLUCOSE CO-TRANSPORTER 2 LEXICON PHARMACEUTICALS, INC. (US) 2008-09-12 WO disclosed
WO-2008042688-A2 PHLORIZIN ANALOGS AS INHIBITORS OF SODIUM GLUCOSE CO-TRANSPORTER 2 LEXICON PHARMACEUTICALS, INC. (US) 2008-04-10 WO disclosed