SCHEMBL2370258

SCHEMBL2370258

CC(C)(C)COc1cc2c(c(F)n1)Oc1ccc(Br)cc1C21CNCC(N)O1

nearest known ligand 0.30

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2371060 0.85 BACE1 (0.34) BACE1
SCHEMBL2370902 0.85 BACE1 (0.47) BACE1
SCHEMBL2370953 0.85 BACE1 (0.47) BACE1
SCHEMBL2370691 0.83 BACE1 (0.34) BACE1
SCHEMBL2370605 0.82 BACE1 (0.34) BACE1
SCHEMBL2371069 0.82 BACE1 (0.34) BACE1
SCHEMBL2371275 0.77 BACE1 (0.37) BACE1
SCHEMBL2371365 0.75 BACE1 (0.35) BACE1
SCHEMBL2371098 0.75 BACE1 (0.35) BACE1
SCHEMBL2370832 0.75 BACE1 (0.35) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-A1 AMINO -DIHYDROOXAZINE AND AMINO - DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA - SECRETASE MODULATORS AND THEIR MEDICAL USE Amgen Inc. (US) 2013-01-23 EP disclosed
WO-2011115928-A1 AMINO -DIHYDROOXAZINE AND AMINO - DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA - SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC. (US) 2011-09-22 WO disclosed