SCHEMBL2370702

SCHEMBL2370702

CNC(=O)c1c(-c2ccc(F)cc2)oc2ccc(-c3cc(C(=O)N(c4ncc(C)s4)C4CC4)ccc3C)cc12

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.57
CYP3A4 P08684 6/20 0.57
KCNH2 Q12809 3/20 0.57
NR1I2 O75469 1/20 0.55
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2370065 0.88 CYP2C8 (0.60) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL2370328 0.88 CYP2C8 (0.60) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL2369508 0.87 CYP2C8 (0.59) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL1919541 0.87 CYP2C8 (0.67) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL1918488 0.87 CYP3A4 (0.61) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL1918981 0.87 CYP3A4 (0.46) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL1919689 0.86 CYP3A4 (0.59) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL2369729 0.85 CYP3A4 (0.60) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL2370004 0.85 CYP2C8 (0.58) CYP2C8CYP3A4KCNH2NR1I2CYP2C9
SCHEMBL1919829 0.85 CYP3A4 (0.66) CYP2C8CYP3A4KCNH2NR1I2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545042-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112191-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed