SCHEMBL23707355

SCHEMBL23707355

Cc1ccc(C#CC(C)(C)C)cc1F

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD5 P21918 1/20 0.36
P2RY6 Q15077 1/20 0.36
GRM5 P41594 3/20 0.34
APP P05067 1/20 0.34
BACE1 P56817 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CYP2D6 P10635 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
FFAR1 O14842 3/20 0.33
FFAR4 Q5NUL3 3/20 0.33
ACHE P22303 1/20 0.32
PTGES2 Q9H7Z7 2/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7851731 0.85 HTT (0.41) KMT2AATM
SCHEMBL17036522 0.85 GRM5 (0.46) DRD5P2RY6GRM5APPBACE1
SCHEMBL17036534 0.84 GRM5 (0.43) DRD5P2RY6GRM5APPBACE1
SCHEMBL31442843 0.83 GRM5 (0.44) GRM5HDAC1HDAC6FFAR1FFAR4
SCHEMBL7859984 0.81 GRM5 (0.43) GRM5APPHDAC1HDAC6FFAR1
SCHEMBL15957582 0.81 DRD5 (0.36) DRD5P2RY6GRM5APPBACE1
SCHEMBL8771565 0.78 CYP1A1 (0.40) GRM5HDAC1HDAC6FFAR1FFAR4
SCHEMBL10018714 0.76 GRM5 (0.44) GRM5HDAC1HDAC6FFAR1FFAR4
SCHEMBL7857769 0.76 GRM5 (0.44) GRM5HDAC1HDAC6FFAR1FFAR4
SCHEMBL3592439 0.74 EPHX2 (0.41) FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3681870-B1 MICROBIOCIDAL QUINOLINE (THIO)CARBOXAMIDE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2021-08-04 EP disclosed