SCHEMBL2371017

SCHEMBL2371017

NC1=NC2(CS1)c1ccccc1Oc1ncccc12

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.36
CTSD P07339 2/20 0.33
KCNH2 Q12809 3/20 0.32
CTSB P07858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2519950 0.81 BACE1 (0.48) BACE1CTSDKCNH2CTSB
SCHEMBL2518831 0.80 BACE1 (0.55) BACE1CTSDKCNH2CTSB
SCHEMBL14629825 0.79 BACE1 (0.31) BACE1CTSD
SCHEMBL2518932 0.78 BACE1 (0.36) BACE1CTSDKCNH2CTSB
SCHEMBL2525174 0.77 BACE1 (0.43) BACE1CTSDKCNH2CTSB
SCHEMBL2522252 0.77 BACE1 (0.36) BACE1CTSDKCNH2
SCHEMBL2517653 0.77 BACE1 (0.56) BACE1CTSDKCNH2CTSB
SCHEMBL2382582 0.74 AHR (0.37) BACE1CTSD
SCHEMBL2522345 0.73 BACE1 (0.33) BACE1
SCHEMBL2524174 0.72 BACE1 (0.36) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547685-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETA - SECRETASE MODULATORS Amgen Inc. (US) 2013-01-23 EP disclosed
WO-2011115938-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETA - SECRETASE MODULATORS AMGEN INC. (US) 2011-09-22 WO disclosed