SCHEMBL2372067

SCHEMBL2372067

CC1(COc2cc3c(cc2F)Oc2ccc(-c4cccc(Cl)c4)cc2[C@@]32COC(N)=N2)COC1

nearest known ligand 0.79

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.79
CTSD P07339 10/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14877619 0.88 BACE1 (1.00) BACE1CTSD
SCHEMBL15510359 0.87 BACE1 (0.84) BACE1CTSD
SCHEMBL15510342 0.87 BACE1 (0.84) BACE1CTSD
SCHEMBL15510349 0.81 BACE1 (0.70) BACE1CTSD
SCHEMBL15510130 0.76 BACE1 (0.70) BACE1CTSD
SCHEMBL2012103 0.76 BACE1 (0.72) BACE1CTSD
SCHEMBL15510016 0.76 BACE1 (0.63) BACE1CTSD
SCHEMBL2384172 0.75 BACE1 (0.60) BACE1CTSD
SCHEMBL14877672 0.75 BACE1 (0.79) BACE1CTSD
SCHEMBL15509794 0.75 BACE1 (0.78) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547685-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETA - SECRETASE MODULATORS Amgen Inc. (US) 2013-01-23 EP disclosed
WO-2011115938-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETA - SECRETASE MODULATORS AMGEN INC. (US) 2011-09-22 WO disclosed