SCHEMBL23723958

SCHEMBL23723958

COC(=O)Cc1ncoc1C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
GAA P10253 2/20 0.38
MAPT P10636 1/20 0.38
HSP90AB1 P08238 1/20 0.38
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
KDM4E B2RXH2 5/20 0.36
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM5B Q9UGL1 1/20 0.35
HSD17B10 Q99714 2/20 0.34
HTT P42858 1/20 0.34
NAMPT P43490 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6712056 0.79 GABRR1 (0.47) SMN1; SMN2GAAMAPTKDM4ERAB9A
SCHEMBL13765710 0.69 GAA (0.39) SMN1; SMN2GAAMAPTHSP90AB1CYP4F2
SCHEMBL2143331 0.68 KDM4E (0.49) SMN1; SMN2MAPTKDM4ERAB9ANPC1
SCHEMBL6712382 0.67
SCHEMBL7882626 0.67 MAPT (0.46) SMN1; SMN2GAAMAPTRAB9ANPC1
SCHEMBL11361086 0.66
SCHEMBL9475115 0.66 MAPT (0.42) SMN1; SMN2GAAMAPTHSP90AB1CYP4F2
SCHEMBL12218698 0.66 DPP4 (0.40) SMN1; SMN2GAAMAPTHSP90AB1CYP4F2
SCHEMBL873517 0.66 NAMPT (0.40) HSP90AB1CYP4F2CYP4A11HSD17B10HTT
SCHEMBL3587690 0.66 SMN1; SMN2 (0.46) SMN1; SMN2GAAMAPTHSP90AB1CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021156439-A1 TRIAZOLE COMPOUNDS AS ADENOSINE RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2021-08-12 WO disclosed
WO-2021156439-A1 TRIAZOLE COMPOUNDS AS ADENOSINE RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2021-08-12 WO disclosed