SCHEMBL23744339

SCHEMBL23744339

C=C[C@@H]1CN(C(=O)Cl)[C@H](C)CN1c1ncc(C(F)(F)F)cn1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
CHRM2 P08172 6/20 0.37
CHRM1 P11229 6/20 0.37
CHRM3 P20309 3/20 0.37
CHRM4 P08173 7/20 0.36
ACACB O00763 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
TIPARP Q7Z3E1 1/20 0.34
CXCR3 P49682 1/20 0.33
HSD11B1 P28845 1/20 0.33
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23744338 0.86 TRPV1 (0.42) SMN1; SMN2CHRM2CHRM1CHRM3CHRM4
SCHEMBL26089136 0.86 TRPV1 (0.42) SMN1; SMN2CHRM2CHRM1CHRM3CHRM4
SCHEMBL26087204 0.75 CHRM2 (0.55) CHRM2CHRM1CHRM3CHRM4
SCHEMBL26087301 0.74 TRPV1 (0.43) CHRM2CHRM1CHRM3CHRM4ACACB
SCHEMBL29165925 0.74 TRPV1 (0.43) CHRM2CHRM1CHRM3CHRM4ACACB
SCHEMBL26089036 0.74 TRPV1 (0.43) CHRM2CHRM1CHRM3CHRM4ACACB
SCHEMBL27233838 0.74 TRPV1 (0.43) CHRM2CHRM1CHRM3CHRM4ACACB
SCHEMBL23728061 0.74 TRPV1 (0.43) CHRM2CHRM1CHRM3CHRM4ACACB
SCHEMBL29165969 0.74 TRPV1 (0.43) CHRM2CHRM1CHRM3CHRM4ACACB
SCHEMBL23744341 0.70 CHRM2 (0.52) SMN1; SMN2CHRM2CHRM1CHRM3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021158698-A1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. (US) 2021-08-12 WO disclosed