SCHEMBL23768947

SCHEMBL23768947

CCOC(=O)c1cn(Cc2ccc(N3CC(C)C(F)(F)C3)nc2C)nc1CCl

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 18/20 0.41
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23768949 0.87 KLKB1 (0.53) KLKB1
SCHEMBL24919158 0.85 KLKB1 (0.52) KLKB1
SCHEMBL23754099 0.84 KLKB1 (0.51) KLKB1
SCHEMBL31357806 0.84 KLKB1 (0.51) KLKB1
SCHEMBL24918819 0.83 KLKB1 (0.48) KLKB1
SCHEMBL23768933 0.81 KLKB1 (0.46) KLKB1
SCHEMBL23769558 0.79 KLKB1 (0.62) KLKB1
SCHEMBL24918413 0.78 KLKB1 (0.46) KLKB1
SCHEMBL24105343 0.77 KLKB1 (0.53) KLKB1
SCHEMBL23769527 0.76 KLKB1 (0.61) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed