SCHEMBL23769205

SCHEMBL23769205

CCOC(=O)c1cnn(Cc2cnc(N3CC4C[C@H]4C3)cc2Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BTK Q06187 10/20 0.47
KLKB1 P03952 8/20 0.40
PIK3CA P42336 1/20 0.36
P2RY12 Q9H244 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843083 1.00 BTK (0.47) BTKKLKB1PIK3CAP2RY12
SCHEMBL18816474 0.90 BTK (0.56) BTKKLKB1PIK3CA
SCHEMBL18815275 0.86 BTK (0.57) BTKKLKB1
SCHEMBL23769232 0.86 BTK (0.47) BTKKLKB1
SCHEMBL23754006 0.83 KLKB1 (0.48) BTKKLKB1
SCHEMBL18795038 0.82 BTK (0.52) BTKKLKB1
SCHEMBL23769685 0.82 BTK (0.39) BTKKLKB1
SCHEMBL23769320 0.81 NOTUM (0.42) BTKKLKB1P2RY12
SCHEMBL23469581 0.80 KLKB1 (0.56) BTKKLKB1
SCHEMBL20540770 0.80 KLKB1 (0.57) BTKKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed