SCHEMBL23769220

SCHEMBL23769220

O=C(O)c1cn(Cc2ccc(N3CC4[C@H](C3)C4(F)F)nc2Br)cn1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 15/20 0.48
RBP4 P02753 1/20 0.33
BTK Q06187 1/20 0.32
USP30 Q70CQ3 1/20 0.32
KDM4E B2RXH2 1/20 0.30
PLA2G4A P47712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843094 1.00 KLKB1 (0.48) KLKB1RBP4BTKUSP30KDM4E
SCHEMBL23769331 0.90 KLKB1 (0.49) KLKB1RBP4BTKUSP30KDM4E
SCHEMBL21736742 0.88 KLKB1 (0.51) KLKB1KDM4E
SCHEMBL23769644 0.88 KLKB1 (0.48) KLKB1RBP4BTKUSP30KDM4E
SCHEMBL23769228 0.87 KLKB1 (0.47) KLKB1RBP4BTK
SCHEMBL31357813 0.87 KLKB1 (0.48) KLKB1KDM4E
SCHEMBL23754036 0.87 KLKB1 (0.48) KLKB1KDM4E
SCHEMBL23768864 0.86 KLKB1 (0.45) KLKB1RBP4BTKUSP30
SCHEMBL23769169 0.86 KLKB1 (0.48) KLKB1RBP4KDM4EPLA2G4A
SCHEMBL23769624 0.86 KLKB1 (0.62) KLKB1RBP4BTKUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed