SCHEMBL23769313

SCHEMBL23769313

CCOC(=O)c1cn(Cc2cnc(N3CC4CC4C3)c(C)c2C)cn1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 8/20 0.48
NOTUM Q6P988 1/20 0.35
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 1/20 0.33
SMYD3 Q9H7B4 1/20 0.32
ALOX15 P16050 1/20 0.32
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31
OPRK1 P41145 1/20 0.31
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
P2RY12 Q9H244 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843030 0.89 KLKB1 (0.62) KLKB1NOTUMALDH1A1MEN1KMT2A
SCHEMBL23769202 0.83 BTK (0.42) KLKB1NOTUMKDM4E
SCHEMBL21736655 0.83 KLKB1 (0.47) KLKB1NOTUM
SCHEMBL23769320 0.81 NOTUM (0.42) KLKB1NOTUMKMT2AP2RY12LMNA
SCHEMBL26309179 0.81 KLKB1 (0.38) KLKB1NOTUMALDH1A1MEN1KMT2A
SCHEMBL30414959 0.81 KLKB1 (0.38) KLKB1NOTUMALDH1A1MEN1KMT2A
SCHEMBL23754197 0.81 KLKB1 (0.38) KLKB1NOTUMALDH1A1MEN1KMT2A
SCHEMBL23769211 0.80 KLKB1 (0.38) KLKB1NOTUMALDH1A1ALOX15KDM4E
SCHEMBL23769281 0.79 KLKB1 (0.45) KLKB1NOTUM
SCHEMBL23754033 0.79 KLKB1 (0.46) KLKB1NOTUMALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed