SCHEMBL23769484

SCHEMBL23769484

CCOC(=O)c1cnn(Cc2ccc(N3CC4C[C@H]4C3)nc2C(C)(C)C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BTK Q06187 6/20 0.46
KLKB1 P03952 13/20 0.44
RET P07949 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843122 1.00 BTK (0.46) BTKKLKB1RET
SCHEMBL23769689 0.90 BTK (0.48) BTKKLKB1
SCHEMBL23843098 0.89 BTK (0.49) BTKKLKB1
SCHEMBL18816600 0.88 BTK (0.58) BTKKLKB1
SCHEMBL21713103 0.86 KLKB1 (0.46) BTKKLKB1RET
SCHEMBL31033231 0.85 KLKB1 (0.57) BTKKLKB1
SCHEMBL20540770 0.85 KLKB1 (0.57) BTKKLKB1
SCHEMBL29906586 0.84 KLKB1 (0.45) BTKKLKB1
SCHEMBL23754342 0.84 KLKB1 (0.45) BTKKLKB1
SCHEMBL23769206 0.84 KLKB1 (0.49) BTKKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed