SCHEMBL23769503

SCHEMBL23769503

C=C1Nc2c(C)cccc2C(c2cccc(F)c2)=NC1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTCH1 P46531 11/20 0.47
NOTCH3 Q9UM47 8/20 0.47
RBPJ Q06330 3/20 0.41
MGAM O43451 1/20 0.36
GAA P10253 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
MAPT P10636 3/20 0.35
ALOX15 P16050 3/20 0.35
ALOX12 P18054 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NFKB1 P19838 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15608508 0.87 NOTCH1 (0.54) NOTCH1NOTCH3RBPJMGAMGAA
SCHEMBL15608509 0.87 NOTCH1 (0.54) NOTCH1NOTCH3RBPJMGAMGAA
SCHEMBL23769413 0.78 NOTCH1 (0.52) NOTCH1NOTCH3RBPJMGAMGAA
SCHEMBL15608401 0.76 NOTCH1 (0.53) NOTCH1NOTCH3RBPJMGAMGAA
SCHEMBL17030708 0.74 NOTCH1 (0.42) NOTCH1NOTCH3RBPJMAPTALOX15
SCHEMBL15622551 0.74 NOTCH1 (0.54) NOTCH1NOTCH3RBPJMEN1KMT2A
SCHEMBL15629462 0.74 NOTCH1 (0.54) NOTCH1NOTCH3RBPJMEN1KMT2A
SCHEMBL15631538 0.74 NOTCH1 (0.58) NOTCH1NOTCH3RBPJ
SCHEMBL15622343 0.74 NOTCH1 (0.45) NOTCH1NOTCH3RBPJBRD4
SCHEMBL15622249 0.74 NOTCH1 (0.58) NOTCH1NOTCH3RBPJ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021163676-A1 METHODS OF PREPARING CHIRAL BENZODIAZEPINONE DERIVATIVES AYALA PHARMACEUTICALS INC. (US) 2021-08-19 WO disclosed